Crystal structure of CDK2 in complex with inhibitor ICEC0942
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Crystal structure of CDK2 in complex with inhibitor ICEC0942 Descriptor: (3R,4R)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-ol, ACETATE ION, Cyclin-dependent kinase 2 Authors: Hazel, P, Freemont, P.S. Deposit date: 2016-05-04 Release date: 2017-02-08 Last modified: 2024-01-10 Method: X-RAY DIFFRACTION (1.94 Å) Cite: Inhibitor Selectivity for Cyclin-Dependent Kinase 7: A Structural, Thermodynamic, and Modelling Study. ChemMedChem, 12, 2017
创建时间:
2016-05-04



