Crystal Structure of Human Kallikrein 5 in complex with GSK144
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Crystal Structure of Human Kallikrein 5 in complex with GSK144 Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 4-[(5-phenyl-1~{H}-imidazol-2-yl)methylamino]-2-(pyridin-3-ylmethoxy)benzenecarboximidamide, ... Authors: Thorpe, J.H. Deposit date: 2019-01-10 Release date: 2019-05-08 Last modified: 2024-11-13 Method: X-RAY DIFFRACTION (1.67 Å) Cite: Evaluation of a crystallographic surrogate for kallikrein 5 in the discovery of novel inhibitors for Netherton syndrome. Acta Crystallogr.,Sect.F, 75, 2019
创建时间:
2019-01-10



