Structure of PI3K gamma with Imidazopyridine inhibitors
收藏Protein Data Bank Japan2024-02-28 更新2026-03-21 收录
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https://pdbj.org/mine/summary/4kzc
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Structure of PI3K gamma with Imidazopyridine inhibitors Descriptor: N-{6-[6-amino-5-(trifluoromethyl)pyridin-3-yl]imidazo[1,2-a]pyridin-2-yl}acetamide, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform, SULFATE ION Authors: Knapp, M.S, Elling, E.A. Deposit date: 2013-05-29 Release date: 2013-07-17 Last modified: 2024-02-28 Method: X-RAY DIFFRACTION (3.25 Å) Cite: Structure guided optimization of a fragment hit to imidazopyridine inhibitors of PI3K. Bioorg.Med.Chem.Lett., 23, 2013
创建时间:
2013-05-29



