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RIP2 Kinase Catalytic Domain complex with 5amino1tertbutyl3(3methoxyphenyl)1H pyrazole4carboxamide.

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Protein Data Bank Japan2024-05-15 更新2026-03-21 收录
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https://pdbj.org/mine/summary/6szj
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资源简介:
RIP2 Kinase Catalytic Domain complex with 5amino1tertbutyl3(3methoxyphenyl)1H pyrazole4carboxamide. Descriptor: 5-amino-1-~{tert}-butyl-3-(3-methoxyphenyl)pyrazole-4-carboxamide, CALCIUM ION, Receptor-interacting serine/threonine-protein kinase 2 Authors: Convery, M.A, Charnley, A.K, Shewchuk, L. Deposit date: 2019-10-02 Release date: 2019-12-04 Last modified: 2024-05-15 Method: X-RAY DIFFRACTION (2.53 Å) Cite: Discovery of Pyrazolocarboxamides as Potent and Selective Receptor Interacting Protein 2 (RIP2) Kinase Inhibitors. Acs Med.Chem.Lett., 10, 2019
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2019-10-02
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