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Crystal structure of the first bromodomain of human BRD4 in complex with DINACICLIB

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Protein Data Bank Japan2023-09-20 更新2026-03-21 收录
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Crystal structure of the first bromodomain of human BRD4 in complex with DINACICLIB Descriptor: 1,2-ETHANEDIOL, 3-[({3-ethyl-5-[(2S)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridinium, Bromodomain-containing protein 4 Authors: Ember, S.W, Zhu, J.-Y, Watts, C, Schonbrunn, E. Deposit date: 2013-12-24 Release date: 2014-03-05 Last modified: 2023-09-20 Method: X-RAY DIFFRACTION (1.55 Å) Cite: Acetyl-lysine Binding Site of Bromodomain-Containing Protein 4 (BRD4) Interacts with Diverse Kinase Inhibitors. Acs Chem.Biol., 9, 2014

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2013-12-24
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