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N-terminal domain of BRD4 with biphenyl-methyamino-dimethylpyridazinone

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Protein Data Bank Japan2024-05-01 更新2026-03-21 收录
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https://pdbj.org/mine/summary/6yqz
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资源简介:
N-terminal domain of BRD4 with biphenyl-methyamino-dimethylpyridazinone Descriptor: 1,2-ETHANEDIOL, 2,4-dimethyl-5-[(2-phenylphenyl)methylamino]pyridazin-3-one, Bromodomain-containing protein 4 Authors: Chung, C. Deposit date: 2020-04-18 Release date: 2021-03-24 Last modified: 2024-05-01 Method: X-RAY DIFFRACTION (1.39 Å) Cite: Application of Atypical Acetyl-lysine Methyl Mimetics in the Development of Selective Inhibitors of the Bromodomain-Containing Protein 7 (BRD7)/Bromodomain-Containing Protein 9 (BRD9) Bromodomains. J.Med.Chem., 63, 2020
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2020-04-18
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