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CRYSTAL STRUCTURE OF THE AGONIST FORM OF GLUCOCORTICOID RECEPTOR

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Protein Data Bank Japan2023-08-16 更新2026-03-21 收录
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CRYSTAL STRUCTURE OF THE AGONIST FORM OF GLUCOCORTICOID RECEPTOR Descriptor: DEXAMETHASONE, Glucocorticoid receptor, Nuclear receptor coactivator 2 Authors: Kauppi, B, Jakob, C, Farnegardh, M, Yang, J, Ahola, H, Alarcon, M, Calles, K, Engstrom, O, Harlan, J, Muchmore, S, Ramqvist, A.-K, Thorell, S, Ohman, L, Greer, J, Gustafsson, J.-A, Carlstedt-Duke, J, Carlquist, M. Deposit date: 2003-05-09 Release date: 2003-07-08 Last modified: 2023-08-16 Method: X-RAY DIFFRACTION (2.7 Å) Cite: The Three-dimensional Structures of Antagonistic and Agonistic Forms of the Glucocorticoid Receptor Ligand-binding Domain: RU-486 INDUCES A TRANSCONFORMATION THAT LEADS TO ACTIVE ANTAGONISM. J.Biol.Chem., 278, 2003
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2003-05-09
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