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Plasmodium vivax PMV-WM06 inhibitor complex

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Protein Data Bank Japan2025-09-10 更新2026-04-19 收录
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Plasmodium vivax PMV-WM06 inhibitor complex Descriptor: (2E,4aR,7aS)-6-[(3M)-3-(2-chlorophenyl)pyridin-2-yl]-7a-(2,5-difluorophenyl)-2-imino-3-methyloctahydro-4H-pyrrolo[3,4-d]pyrimidin-4-one, 1,2-ETHANEDIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, ... Authors: Hodder, A.N, Scally, S.W, Czabotar, P.E, Cowman, A.F. Deposit date: 2023-08-25 Release date: 2024-08-28 Last modified: 2025-09-10 Method: X-RAY DIFFRACTION (2.59 Å) Cite: Structure-activity analysis of imino-pyrimidinone-fused pyrrolidines aids the development of dual plasmepsin V and plasmepsin X inhibitors. Febs J., 292, 2025

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2023-08-25
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