Crystal structure of compound 8 bound to TAK1-TAB
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Crystal structure of compound 8 bound to TAK1-TAB Descriptor: (1E)-1-[5-TERT-BUTYL-2-(3-FLUOROPHENYL)-1H-PYRAZOL-3-YLIDENE]-3-(4-PYRIDIN-3-YLOXYPHENYL)UREA, MITOGEN-ACTIVATED PROTEIN KINASE KINASE KINASE 7, TGF-BETA-ACTIVATED KINASE 1 AND MAP3K7-BINDING PROTEIN 1 Authors: Brown, D.G, Phillips, C. Deposit date: 2011-05-17 Release date: 2012-05-23 Last modified: 2023-12-20 Method: X-RAY DIFFRACTION (2.49 Å) Cite: The Discovery and Synthesis of Selective Dfg-Out Tak-1 Inhibitors To be Published
创建时间:
2011-05-17



