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Crystal Structure of Anaplastic Lymphoma Kinase Complexed with LDK378

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Protein Data Bank Japan2023-09-20 更新2026-03-21 收录
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Crystal Structure of Anaplastic Lymphoma Kinase Complexed with LDK378 Descriptor: 5-chloro-N~2~-[5-methyl-4-(piperidin-4-yl)-2-(propan-2-yloxy)phenyl]-N~4~-[2-(propan-2-ylsulfonyl)phenyl]pyrimidine-2,4-diamine, ALK tyrosine kinase receptor, GLYCEROL Authors: Lee, C.C, Spraggon, G. Deposit date: 2013-09-04 Release date: 2014-04-09 Last modified: 2023-09-20 Method: X-RAY DIFFRACTION (2.01 Å) Cite: The ALK Inhibitor Ceritinib Overcomes Crizotinib Resistance in Non-Small Cell Lung Cancer. Cancer Discov, 4, 2014
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2013-09-04
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