five

Crystal Structure of BAZ2A bromodomain in complex with 1,3-dimethyl-benzimidazolone compound 1

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Protein Data Bank Japan2024-01-17 更新2026-03-21 收录
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Crystal Structure of BAZ2A bromodomain in complex with 1,3-dimethyl-benzimidazolone compound 1 Descriptor: Bromodomain adjacent to zinc finger domain protein 2A, ~{N}-[(4-fluorophenyl)methyl]-1,3,6-trimethyl-2-oxidanylidene-benzimidazole-5-sulfonamide Authors: Lolli, G, Dalle Vedove, A, Marchand, J.-R, Caflisch, A. Deposit date: 2017-08-15 Release date: 2017-09-13 Last modified: 2024-01-17 Method: X-RAY DIFFRACTION (2.4 Å) Cite: Discovery of Inhibitors of Four Bromodomains by Fragment-Anchored Ligand Docking. J Chem Inf Model, 57, 2017
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2017-08-15
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