Crystal structure of Retinoic Acid Receptor alpha (RXRA) in complexed with S169 inhibitor
收藏Protein Data Bank Japan2024-01-31 更新2026-03-21 收录
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Crystal structure of Retinoic Acid Receptor alpha (RXRA) in complexed with S169 inhibitor Descriptor: 3-(5-(3,5-bis(trifluoromethyl)phenyl)-4-phenyloxazol-2-yl)propanoic acid, Nuclear receptor coactivator 2, Retinoic acid receptor RXR-alpha Authors: Ni, X, Chaikuad, A, Schierle, S, Merk, D, Knapp, S, Structural Genomics Consortium (SGC) Deposit date: 2020-12-14 Release date: 2021-02-10 Last modified: 2024-01-31 Method: X-RAY DIFFRACTION (2.05 Å) Cite: Oxaprozin Analogues as Selective RXR Agonists with Superior Properties and Pharmacokinetics. J.Med.Chem., 64, 2021
创建时间:
2020-12-14



