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Endothiapepsin complex with renin inhibitor MERCK-KGAA-EMD61395

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Protein Data Bank Japan2024-10-23 更新2026-03-21 收录
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https://pdbj.org/mine/summary/1e81
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Endothiapepsin complex with renin inhibitor MERCK-KGAA-EMD61395 Descriptor: (2S)-1-{[(2R)-1-{[(2S,3S)-1-cyclohexyl-3-hydroxy-4-(2-oxopyridin-1(2H)-yl)butan-2-yl]amino}-3-(methylsulfanyl)-1-oxopropan-2-yl]amino}-1-oxo-3-phenylpropan-2-yl 4-aminopiperidine-1-carboxylate, ENDOTHIAPEPSIN Authors: Read, J.A, Cooper, J.B, Toldo, L, Rippmann, F, Raddatz, P. Deposit date: 2000-09-15 Release date: 2000-10-19 Last modified: 2024-10-23 Method: X-RAY DIFFRACTION (2.05 Å) Cite: Refinement of Four Endothiapepsin Inhibitor Complexes. Crystallographic Studies of Cytochrome Ch from Methylobacterium Extorquens and Inhibitor Complexes of Aspartic Proteinases. Thesis, 1999
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2000-09-15
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