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Non peptide agonist PF-06882961, bound to Glucagon-Like peptide-1 (GLP-1) Receptor

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Protein Data Bank Japan2025-05-28 更新2026-03-21 收录
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https://pdbj.org/mine/summary/6x1a
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Non peptide agonist PF-06882961, bound to Glucagon-Like peptide-1 (GLP-1) Receptor Descriptor: 2-[(4-{6-[(4-cyano-2-fluorophenyl)methoxy]pyridin-2-yl}piperidin-1-yl)methyl]-1-{[(2S)-oxetan-2-yl]methyl}-1H-benzimidazole-6-carboxylic acid, Glucagon-like peptide 1 receptor, Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2, ... Authors: Belousoff, M.J, Zhang, X, Danev, R. Deposit date: 2020-05-18 Release date: 2020-09-09 Last modified: 2025-05-28 Method: ELECTRON MICROSCOPY (2.5 Å) Cite: Differential GLP-1R Binding and Activation by Peptide and Non-peptide Agonists. Mol.Cell, 80, 2020
创建时间:
2020-05-18
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