BRD4_BD2_A-1497627
收藏Protein Data Bank Japan2024-04-03 更新2026-03-21 收录
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https://pdbj.org/mine/summary/5uex
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BRD4_BD2_A-1497627 Descriptor: 17-{[ethyl(dihydroxy)-lambda~4~-sulfanyl]amino}-11,13-difluoro-2-methyl-6,7,8,9-tetrahydrodibenzo[4,5:7,8][1,6]dioxacyclododecino[3,2-c]pyridin-3(2H)-one, Bromodomain-containing protein 4 Authors: Park, C.H. Deposit date: 2017-01-03 Release date: 2017-05-10 Last modified: 2024-04-03 Method: X-RAY DIFFRACTION (2.29 Å) Cite: Fragment-Based, Structure-Enabled Discovery of Novel Pyridones and Pyridone Macrocycles as Potent Bromodomain and Extra-Terminal Domain (BET) Family Bromodomain Inhibitors. J. Med. Chem., 60, 2017
创建时间:
2017-01-03



