遇见数据集

MLL1 SET N3861I/Q3867L bound to inhibitor 12 (TC-5140)

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Protein Data Bank Japan2023-10-11 更新2026-03-21 收录
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MLL1 SET N3861I/Q3867L bound to inhibitor 12 (TC-5140) Descriptor: 5'-{[(3S)-3-amino-3-carboxypropyl]({1-[(3-chlorophenyl)methyl]azetidin-3-yl}methyl)amino}-5'-deoxyadenosine, Histone-lysine N-methyltransferase, ZINC ION Authors: Petrunak, E.M, Stuckey, J.A. Deposit date: 2019-09-09 Release date: 2020-07-01 Last modified: 2023-10-11 Method: X-RAY DIFFRACTION (2.1 Å) Cite: Discovery of Potent Small-Molecule Inhibitors of MLL Methyltransferase. Acs Med.Chem.Lett., 11, 2020

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2019-09-09
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