five

Glycogen Synthase Kinase 3 beta Complexed with BRD0705

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Protein Data Bank Japan2024-10-23 更新2026-03-21 收录
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Glycogen Synthase Kinase 3 beta Complexed with BRD0705 Descriptor: (4~{S})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-one, Glycogen synthase kinase-3 beta Authors: Lakshminarasimhan, D, White, A, Nadupalli, A, Suto, R.K. Deposit date: 2016-07-04 Release date: 2018-03-14 Last modified: 2024-10-23 Method: X-RAY DIFFRACTION (2.6 Å) Cite: Exploiting an Asp-Glu "switch" in glycogen synthase kinase 3 to design paralog-selective inhibitors for use in acute myeloid leukemia. Sci Transl Med, 10, 2018
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2016-07-04
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