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Structure of the human GluN1/GluN2A LBD in complex with GNE0723

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Protein Data Bank Japan2024-11-06 更新2026-03-21 收录
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Structure of the human GluN1/GluN2A LBD in complex with GNE0723 Descriptor: (1~{R},2~{R})-2-[7-[[5-chloranyl-3-(trifluoromethyl)pyrazol-1-yl]methyl]-5-oxidanylidene-2-(trifluoromethyl)-[1,3]thiazolo[3,2-a]pyrimidin-3-yl]cyclopropane-1-carbonitrile, ACETATE ION, GLUTAMIC ACID, ... Authors: Wallweber, H.J.A, Lupardus, P.J. Deposit date: 2016-06-08 Release date: 2016-07-13 Last modified: 2024-11-06 Method: X-RAY DIFFRACTION (2.44 Å) Cite: Discovery of GluN2A-Selective NMDA Receptor Positive Allosteric Modulators (PAMs): Tuning Deactivation Kinetics via Structure-Based Design. J. Med. Chem., 59, 2016
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2016-06-08
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