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Human Deoxyhypusine Synthase Fragment Screening Campaign - ligand VT00223

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Protein Data Bank Japan2026-02-18 更新2026-04-19 收录
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Human Deoxyhypusine Synthase Fragment Screening Campaign - ligand VT00223 Descriptor: (4R)-2-METHYLPENTANE-2,4-DIOL, 2-fluoranyl-~{N},~{N}-dimethyl-benzenesulfonamide, Deoxyhypusine synthase, ... Authors: Wilk, P, Wator-Wilk, E, Krojer, T, Grudnik, P. Deposit date: 2025-02-15 Release date: 2026-01-21 Last modified: 2026-02-18 Method: X-RAY DIFFRACTION (1.35 Å) Cite: Crystallographic fragment screening supports tool compound discovery and reveals conformational flexibility in human deoxyhypusine synthase. Commun Chem, 9, 2026

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2025-02-15
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