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BAZ2A bromodomain in complex with acetylpyrrole derivative compound 109

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Protein Data Bank Japan2024-01-31 更新2026-04-19 收录
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BAZ2A bromodomain in complex with acetylpyrrole derivative compound 109 Descriptor: (2~{R})-1-[4-(4-ethanoyl-3-ethyl-5-methyl-1~{H}-pyrrol-2-yl)-1,3-thiazol-2-yl]-~{N}-(4-oxidanylbutyl)piperazine-2-carboxamide, Bromodomain adjacent to zinc finger domain protein 2A, MAGNESIUM ION Authors: Dalle Vedove, A, Cazzanelli, G, Caflisch, A, Lolli, G. Deposit date: 2022-01-29 Release date: 2022-09-28 Last modified: 2024-01-31 Method: X-RAY DIFFRACTION (2.25 Å) Cite: Identification of a BAZ2A-Bromodomain Hit Compound by Fragment Growing. Acs Med.Chem.Lett., 13, 2022

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2022-01-29
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