Crystal structure of DYRK1A complexed with KuFal319 (compound 11)
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Crystal structure of DYRK1A complexed with KuFal319 (compound 11) Descriptor: 4-chloranyl-5~{H}-cyclohepta[b]indol-10-one, Dual specificity tyrosine-phosphorylation-regulated kinase 1A, SULFATE ION, ... Authors: Chaikuad, A, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Kunick, C, Knapp, S, Structural Genomics Consortium (SGC) Deposit date: 2019-10-18 Release date: 2019-12-04 Last modified: 2024-11-13 Method: X-RAY DIFFRACTION (2.8 Å) Cite: [ b ]-Annulated Halogen-Substituted Indoles as Potential DYRK1A Inhibitors. Molecules, 24, 2019
创建时间:
2019-10-18



