BRD4(BD1) complexed with 3219
收藏Protein Data Bank Japan2024-11-06 更新2026-03-21 收录
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https://pdbj.org/mine/summary/6czu
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BRD4(BD1) complexed with 3219 Descriptor: 1,2-ETHANEDIOL, 5-(3,5-dimethyl-1,2-oxazol-4-yl)-1-({4-[(1R)-1-hydroxyethyl]phenyl}methyl)pyridin-2(1H)-one, Bromodomain-containing protein 4, ... Authors: Lakshminarasimhan, D, White, A, Suto, R.K. Deposit date: 2018-04-09 Release date: 2018-09-26 Last modified: 2024-11-06 Method: X-RAY DIFFRACTION (1.47 Å) Cite: Design and Characterization of Novel Covalent Bromodomain and Extra-Terminal Domain (BET) Inhibitors Targeting a Methionine. J. Med. Chem., 61, 2018
创建时间:
2018-04-09



