Crystal Structure of human Serine/Threonine Kinase 17B (STK17B) in complex with Quercetin
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Crystal Structure of human Serine/Threonine Kinase 17B (STK17B) in complex with Quercetin Descriptor: 3,5,7,3',4'-PENTAHYDROXYFLAVONE, Serine/threonine-protein kinase 17B Authors: Ugochukwu, E, Soundararajan, M, Rellos, P, Fedorov, O, Phillips, C, Wang, J, Hapka, E, Filippakopoulos, P, Chaikuad, A, Pike, A.C.W, Carpenter, L, Vollmar, M, von Delft, F, Bountra, C, Arrowsmith, C.H, Weigelt, J, Edwards, A, Knapp, S, Structural Genomics Consortium (SGC) Deposit date: 2010-01-29 Release date: 2010-03-16 Last modified: 2023-09-06 Method: X-RAY DIFFRACTION (2.29 Å) Cite: A Chemical Probe for Dark Kinase STK17B Derives Its Potency and High Selectivity through a Unique P-Loop Conformation. J.Med.Chem., 63, 2020
创建时间:
2010-01-29



