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EthR from Mycobacterium tuberculosis in complex with compound BDM14950

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Protein Data Bank Japan2024-02-21 更新2026-03-21 收录
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https://pdbj.org/mine/summary/3o8h
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EthR from Mycobacterium tuberculosis in complex with compound BDM14950 Descriptor: 4-iodo-N-[(1-{2-oxo-2-[4-(3-thiophen-2-yl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]ethyl}-1H-1,2,3-triazol-4-yl)methyl]benzenesulfonamide, Transcriptional Regulatory Repressor protein (TETR-Family) EthR Authors: Willand, N, Desroses, M, Toto, P, Diri, B, Lens, Z, Villeret, V, Rucktooa, P, Locht, C, Baulard, A, Deprez, B. Deposit date: 2010-08-03 Release date: 2010-09-01 Last modified: 2024-02-21 Method: X-RAY DIFFRACTION (1.9 Å) Cite: Exploring drug target flexibility using in situ click chemistry: application to a mycobacterial transcriptional regulator. Acs Chem.Biol., 5, 2010
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2010-08-03
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