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Nek2 kinase covalently bound to 2-arylamino-6-ethynylpurine inhibitor 66

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Protein Data Bank Japan2024-10-09 更新2026-03-21 收录
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https://pdbj.org/mine/summary/6sgh
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Nek2 kinase covalently bound to 2-arylamino-6-ethynylpurine inhibitor 66 Descriptor: 2-[4-[(6-ethenyl-9~{H}-purin-2-yl)amino]phenyl]ethanamide, Serine/threonine-protein kinase Nek2 Authors: Richards, M.W, Mas-Droux, C.P, Bayliss, R. Deposit date: 2019-08-04 Release date: 2020-06-17 Last modified: 2024-10-09 Method: X-RAY DIFFRACTION (3 Å) Cite: 2-Arylamino-6-ethynylpurines are cysteine-targeting irreversible inhibitors of Nek2 kinase. Rsc Med Chem, 11, 2020
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2019-08-04
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