Crystal structure of MLLT1 (ENL) YEATS domain in complexed with benzimidazole-amide derivative 6
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Crystal structure of MLLT1 (ENL) YEATS domain in complexed with benzimidazole-amide derivative 6 Descriptor: 1,2-ETHANEDIOL, 4-iodanyl-~{N}-[2-(piperidin-1-ylmethyl)-3~{H}-benzimidazol-5-yl]benzamide, Protein ENL Authors: Chaikuad, A, Heidenreich, D, Moustakim, M, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Fedorov, O, Brennan, P.E, Knapp, S, Structural Genomics Consortium (SGC) Deposit date: 2019-10-04 Release date: 2019-11-06 Last modified: 2024-01-24 Method: X-RAY DIFFRACTION (1.9 Å) Cite: Structural Insights into Interaction Mechanisms of Alternative Piperazine-urea YEATS Domain Binders in MLLT1. Acs Med.Chem.Lett., 10, 2019
创建时间:
2019-10-04



