遇见数据集

Bromodomain and Extra-terminal Domain (BET) BRD4

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Protein Data Bank Japan2024-11-20 更新2026-04-19 收录
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Bromodomain and Extra-terminal Domain (BET) BRD4 Descriptor: 7-[2-fluoranyl-3-(1,3,5-trimethylpyrazol-4-yl)phenyl]-1~{H}-imidazo[4,5-b]pyridine, Bromodomain-containing protein 4 Authors: Cao, D, Zhiyan, D, Xiong, B. Deposit date: 2023-02-13 Release date: 2023-10-04 Last modified: 2024-11-20 Method: X-RAY DIFFRACTION (1.57 Å) Cite: Discovery of 1 H -Imidazo[4,5- b ]pyridine Derivatives as Potent and Selective BET Inhibitors for the Management of Neuropathic Pain. J.Med.Chem., 66, 2023

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2023-02-13
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