Crystal Structure of the first bromodomain of human BRD4 in complex with the inhibitor ZL0590
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Crystal Structure of the first bromodomain of human BRD4 in complex with the inhibitor ZL0590 Descriptor: Bromodomain-containing protein 4, DIMETHYL SULFOXIDE, N-[4-({(2S)-2-[(morpholin-4-yl)methyl]pyrrolidin-1-yl}sulfonyl)phenyl]-N'-[4-(trifluoromethyl)phenyl]urea Authors: Leonard, P.G, Joseph, S. Deposit date: 2019-08-14 Release date: 2020-08-19 Last modified: 2023-10-11 Method: X-RAY DIFFRACTION (1.43 Å) Cite: Discovery, X-ray Crystallography, and Anti-inflammatory Activity of Bromodomain-containing Protein 4 (BRD4) BD1 Inhibitors Targeting a Distinct New Binding Site J. Med. Chem., 2022
创建时间：
2019-08-14
