five

p110delta/p85alpha with taselisib (GDC-0032)

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Protein Data Bank Japan2023-10-04 更新2026-03-21 收录
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https://pdbj.org/mine/summary/5t8f
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p110delta/p85alpha with taselisib (GDC-0032) Descriptor: 2-methyl-2-(4-{2-[3-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-1H-pyrazol-1-yl)propanamide, Phosphatidylinositol 3-kinase regulatory subunit alpha, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform Authors: Moertl, M, Steinbacher, S, Eigenbrot, C. Deposit date: 2016-09-07 Release date: 2017-01-11 Last modified: 2023-10-04 Method: X-RAY DIFFRACTION (2.91 Å) Cite: Structure-Based Design of Tricyclic NF-kappa B Inducing Kinase (NIK) Inhibitors That Have High Selectivity over Phosphoinositide-3-kinase (PI3K). J. Med. Chem., 60, 2017
创建时间:
2016-09-07
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