five

KIT kinase domain mutant D816H in complex with sunitinib

收藏
Protein Data Bank Japan2024-04-03 更新2026-03-21 收录
下载链接:
https://pdbj.org/mine/summary/3g0f
下载链接
链接失效反馈
官方服务:
资源简介:
KIT kinase domain mutant D816H in complex with sunitinib Descriptor: Mast/stem cell growth factor receptor, N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fluoro-2-oxo-1,2-dihydro-3H-indol-3-ylidene)methyl]-2,4-dimethyl-1H-pyrrole-3-carbo xamide, SULFATE ION Authors: Gajiwala, K.S, Wu, J.C, Lunney, E.A, Demetri, G.D. Deposit date: 2009-01-27 Release date: 2009-02-24 Last modified: 2024-04-03 Method: X-RAY DIFFRACTION (2.6 Å) Cite: KIT kinase mutants show unique mechanisms of drug resistance to imatinib and sunitinib in gastrointestinal stromal tumor patients. Proc.Natl.Acad.Sci.USA, 106, 2009
创建时间:
2009-01-27
二维码
社区交流群
二维码
科研交流群
商业服务