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BROMODOMAIN OF HUMAN TAF1 (2) WITH naphthyridinone compound

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Protein Data Bank Japan2024-01-31 更新2026-04-19 收录
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https://pdbj.org/mine/summary/7p4s
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资源简介:
BROMODOMAIN OF HUMAN TAF1 (2) WITH naphthyridinone compound Descriptor: 8-[[1-(3-azanylpropyl)piperidin-4-yl]amino]-5-[5-(hydroxymethyl)pyridin-3-yl]-3-methyl-1~{H}-1,7-naphthyridin-2-one, Isoform 2a of Transcription initiation factor TFIID subunit 1 Authors: Chung, C. Deposit date: 2021-07-13 Release date: 2021-10-13 Last modified: 2024-01-31 Method: X-RAY DIFFRACTION (2.17 Å) Cite: Optimization of Naphthyridones into Selective TATA-Binding Protein Associated Factor 1 (TAF1) Bromodomain Inhibitors. Acs Med.Chem.Lett., 12, 2021
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2021-07-13
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