five

ARUK3000263 complex with Notum

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Protein Data Bank Japan2024-10-16 更新2026-03-21 收录
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https://pdbj.org/mine/summary/6zvl
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资源简介:
ARUK3000263 complex with Notum Descriptor: 1,2-ETHANEDIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, 5-[4-chloranyl-3-(trifluoromethyl)phenyl]-3~{H}-1,3,4-oxadiazol-2-one, ... Authors: Zhao, Y, Ruza, R. Deposit date: 2020-07-24 Release date: 2020-11-11 Last modified: 2024-10-16 Method: X-RAY DIFFRACTION (1.3 Å) Cite: 5-Phenyl-1,3,4-oxadiazol-2(3 H )-ones Are Potent Inhibitors of Notum Carboxylesterase Activity Identified by the Optimization of a Crystallographic Fragment Screening Hit. J.Med.Chem., 63, 2020
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2020-07-24
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