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N-TERMINAL BROMODOMAIN OF HUMAN BRD4 WITH IBET-295

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Protein Data Bank Japan2024-05-08 更新2026-03-21 收录
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资源简介:
N-TERMINAL BROMODOMAIN OF HUMAN BRD4 WITH IBET-295 Descriptor: 1,2-ETHANEDIOL, BROMODOMAIN-CONTAINING PROTEIN 4, propan-2-yl N-[(2S,4R)-1-ethanoyl-2-methyl-6-[4-(methylaminomethyl)phenyl]-3,4-dihydro-2H-quinolin-4-yl]carbamate Authors: Chung, C, Atkinson, S. Deposit date: 2014-01-13 Release date: 2014-12-24 Last modified: 2024-05-08 Method: X-RAY DIFFRACTION (1.6 Å) Cite: The Structure Based Design of Dual Hdac/Bet Inhibitors as Novel Epigenetic Probes. Medchemcomm, 5, 2014
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2014-01-13
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