ERK2 covelently bound to RU60 cyclohexenone based inhibitor
收藏Protein Data Bank Japan2024-10-16 更新2026-04-19 收录
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ERK2 covelently bound to RU60 cyclohexenone based inhibitor Descriptor: AMP PHOSPHORAMIDATE, Mitogen-activated protein kinase 1, ~{O}3-~{tert}-butyl ~{O}1-methyl (1~{R},3~{S})-1-methyl-4-oxidanylidene-cyclohexane-1,3-dicarboxylate Authors: Sok, P, Poti, A, Remenyi, A, Gogl, G. Deposit date: 2023-07-13 Release date: 2024-07-24 Last modified: 2024-10-16 Method: X-RAY DIFFRACTION (1.9 Å) Cite: Targeting a key protein-protein interaction surface on mitogen-activated protein kinases by a precision-guided warhead scaffold. Nat Commun, 15, 2024
创建时间:
2023-07-13



