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Structure of GPR61 bound to inverse agonist compound 15

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Protein Data Bank Japan2026-04-01 更新2026-05-23 收录
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Structure of GPR61 bound to inverse agonist compound 15 Descriptor: Fab24 BAK5 heavy chain, Fab24 BAK5 light chain, G-protein coupled receptor 61,Soluble cytochrome b562, ... Authors: Lees, J.A, Dias, J.M, Han, S. Deposit date: 2025-09-26 Release date: 2026-03-25 Last modified: 2026-04-01 Method: ELECTRON MICROSCOPY (3.08 Å) Cite: Discovery of Potent and Brain-Penetrant Inverse Agonists for GPR61, an Orphan G Protein-Coupled Receptor. J.Med.Chem., 69, 2026

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2025-09-26
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