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Fragment based discovery of JAK-2 inhibitors

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Protein Data Bank Japan2024-10-16 更新2026-03-21 收录
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Fragment based discovery of JAK-2 inhibitors Descriptor: 4-(3-amino-1H-indazol-5-yl)-N-tert-butylbenzenesulfonamide, Tyrosine-protein kinase JAK2 Authors: Antonysamy, S, Fang, W, Hirst, G, Park, F, Russell, M, Smyth, L, Sprengeler, P, Stappenbeck, F, Steensma, R, Thompson, D.A, Wilson, M, Wong, M, Zhang, A, Zhang, F. Deposit date: 2008-08-14 Release date: 2008-10-14 Last modified: 2024-10-16 Method: X-RAY DIFFRACTION (1.8 Å) Cite: Fragment-based discovery of JAK-2 inhibitors. Bioorg.Med.Chem.Lett., 19, 2009

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2008-08-14
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