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Crystal structure of RORc in complex with a phenyl sulfonamide agonist

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Protein Data Bank Japan2023-12-27 更新2026-03-21 收录
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Crystal structure of RORc in complex with a phenyl sulfonamide agonist Descriptor: N-[4-(4-acetylpiperazin-1-yl)-2-fluorobenzyl]-N-cyclobutylbenzenesulfonamide, Nuclear receptor ROR-gamma, RHKILHRLLQEGSPS Authors: Kiefer, J.R, Wallweber, H.A, de Leon Boenig, G, Hymowitz, S.G. Deposit date: 2014-10-18 Release date: 2015-01-14 Last modified: 2023-12-27 Method: X-RAY DIFFRACTION (2.202 Å) Cite: Minor Structural Change to Tertiary Sulfonamide RORc Ligands Led to Opposite Mechanisms of Action. Acs Med.Chem.Lett., 6, 2015
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2014-10-18
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