five

Human kallikrein 7 in complex with 1,4-diazepane-7-one 1-acetamide derivative

收藏
Protein Data Bank Japan2024-10-09 更新2026-03-21 收录
下载链接:
https://pdbj.org/mine/summary/5yjk
下载链接
链接失效反馈
官方服务:
资源简介:
Human kallikrein 7 in complex with 1,4-diazepane-7-one 1-acetamide derivative Descriptor: (R)-2-(6-(5-chloro-2-methoxybenzyl)-3-(2,2-dimethylhydrazono)-7-oxo-1,4-diazepan-1-yl)-N-(3-(methylsulfonyl)phenyl)acetamide, CHLORIDE ION, Kallikrein-7 Authors: Sugawara, H. Deposit date: 2017-10-11 Release date: 2017-12-06 Last modified: 2024-10-09 Method: X-RAY DIFFRACTION (2.4 Å) Cite: Discovery and structure-activity relationship study of 1,3,6-trisubstituted 1,4-diazepane-7-ones as novel human kallikrein 7 inhibitors Bioorg. Med. Chem. Lett., 27, 2017
创建时间:
2017-10-11
二维码
社区交流群
二维码
科研交流群
商业服务