Crystal structure of p38alpha C162S in complex with SB20358 and CAS 2094667-81-7 (behind catalytic site; Y35 in), P 21 21 21
收藏Protein Data Bank Japan2024-02-07 更新2026-04-19 收录
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Crystal structure of p38alpha C162S in complex with SB20358 and CAS 2094667-81-7 (behind catalytic site; Y35 in), P 21 21 21 Descriptor: 4-[4-(4-fluorophenyl)-2-[4-[methyl(oxidanyl)-$l^{3}-sulfanyl]phenyl]-1~{H}-imidazol-5-yl]pyridine, Mitogen-activated protein kinase 14, N-(2-cyclobutyl-1H-1,3-benzodiazol-5-yl)benzenesulfonamide Authors: Baginski, B, Pous, J, Gonzalez, L, Macias, M.J, Nebreda, A.R. Deposit date: 2022-03-11 Release date: 2023-06-14 Last modified: 2024-02-07 Method: X-RAY DIFFRACTION (2.25 Å) Cite: Characterization of p38 alpha autophosphorylation inhibitors that target the non-canonical activation pathway. Nat Commun, 14, 2023
创建时间:
2022-03-11



