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Back pocket flexibility provides group-II PAK selectivity for type 1 kinase inhibitors

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Protein Data Bank Japan2024-11-20 更新2026-03-21 收录
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Back pocket flexibility provides group-II PAK selectivity for type 1 kinase inhibitors Descriptor: PF-3758309, Serine/threonine-protein kinase PAK 1 Authors: Rouge, L, Tam, C, Wang, W. Deposit date: 2013-12-14 Release date: 2014-02-12 Last modified: 2024-11-20 Method: X-RAY DIFFRACTION (2.4 Å) Cite: Back Pocket Flexibility Provides Group II p21-Activated Kinase (PAK) Selectivity for Type I 1/2 Kinase Inhibitors. J.Med.Chem., 57, 2014

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2013-12-14
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