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Crystal Structure of PPARgamma bound to partial agonist MRL24

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Protein Data Bank Japan2023-08-30 更新2026-03-21 收录
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Crystal Structure of PPARgamma bound to partial agonist MRL24 Descriptor: (2S)-2-(3-{[1-(4-METHOXYBENZOYL)-2-METHYL-5-(TRIFLUOROMETHOXY)-1H-INDOL-3-YL]METHYL}PHENOXY)PROPANOIC ACID, Peroxisome Proliferator-Activated Receptor gamma Authors: Bruning, J.B, Nettles, K.W. Deposit date: 2007-06-01 Release date: 2007-10-23 Last modified: 2023-08-30 Method: X-RAY DIFFRACTION (2.3 Å) Cite: Partial Agonists Activate PPARgamma Using a Helix 12 Independent Mechanism Structure, 15, 2007

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2007-06-01
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