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REPLACE: A strategy for Iterative Design of Cyclin Binding Groove Inhibitors

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Protein Data Bank Japan2023-12-13 更新2026-03-21 收录
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REPLACE: A strategy for Iterative Design of Cyclin Binding Groove Inhibitors Descriptor: CELL DIVISION PROTEIN KINASE 2, CYCLIN-A2, N~2~-{[1-(4-CHLOROPHENYL)-5-METHYL-1H-1,2,4-TRIAZOL-3-YL]CARBONYL}-N~5~-(DIAMINOMETHYLIDENE)-L-ORNITHYL-L-LEUCYL-L-ISOLEUCYL-4-FLUORO-L-PHENYLALANINAMIDE Authors: Andrews, M.J, Kontopidis, G, McInnes, C, Plater, A, Innes, L, Cowan, A, Jewsbury, P, Fischer, P.M. Deposit date: 2007-05-31 Release date: 2008-01-29 Last modified: 2023-12-13 Method: X-RAY DIFFRACTION (2.6 Å) Cite: Replace: A Strategy for Iterative Design of Cyclin- Binding Groove Inhibitors Chembiochem, 7, 2006
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2007-05-31
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