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Crystal structure of BTK kinase domain complexed with R406

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Protein Data Bank Japan2023-09-06 更新2026-03-21 收录
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Crystal structure of BTK kinase domain complexed with R406 Descriptor: 6-({5-fluoro-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}amino)-2,2-dimethyl-2H-pyrido[3,2-b][1,4]oxazin-3(4H)-one, Tyrosine-protein kinase BTK Authors: Kuglstatter, A, Wong, A. Deposit date: 2010-11-08 Release date: 2011-01-12 Last modified: 2023-09-06 Method: X-RAY DIFFRACTION (2.55 Å) Cite: Insights into the conformational flexibility of Bruton's tyrosine kinase from multiple ligand complex structures. Protein Sci., 20, 2011
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2010-11-08
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