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Crystal structure of MYST acetyltransferase domain in complex with inhibitor CTX-124143

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Protein Data Bank Japan2024-11-20 更新2026-03-21 收录
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Crystal structure of MYST acetyltransferase domain in complex with inhibitor CTX-124143 Descriptor: 2-fluoro-N'-[(naphthalen-2-yl)sulfonyl]benzohydrazide, GLYCEROL, Histone acetyltransferase KAT8, ... Authors: Hermans, S.J, Chung, M.C, Parker, M.W, Thomas, T, Baell, J.B. Deposit date: 2019-04-09 Release date: 2019-07-03 Last modified: 2024-11-20 Method: X-RAY DIFFRACTION (1.7 Å) Cite: Discovery of Benzoylsulfonohydrazides as Potent Inhibitors of the Histone Acetyltransferase KAT6A. J.Med.Chem., 62, 2019
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2019-04-09
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