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Crystal structure of HDAC8-inhibitor complex

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Protein Data Bank Japan2023-12-13 更新2026-03-21 收录
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Crystal structure of HDAC8-inhibitor complex Descriptor: (2R)-N~8~-HYDROXY-2-{[(5-METHOXY-2-METHYL-1H-INDOL-3-YL)ACETYL]AMINO}-N~1~-[2-(2-PHENYL-1H-INDOL-3-YL)ETHYL]OCTANEDIAMIDE, HISTONE DEACETYLASE 8, POTASSIUM ION, ... Authors: Di Marco, S, Vannini, A, Volpari, C, Gallinari, P, Jones, P, Mattu, M, Carfi, A, Defrancesco, R, Steinkuhler, C. Deposit date: 2007-07-10 Release date: 2007-09-04 Last modified: 2023-12-13 Method: X-RAY DIFFRACTION (2.25 Å) Cite: Substrate Binding to Histone Deacetylases as Revealed by Crystal Structure of Hdac8-Substrate Complex Embo Rep., 8, 2007
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2007-07-10
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