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X-Ray structure of Human Deoxycytidine Kinase in complex with an inhibitor

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Protein Data Bank Japan2023-09-06 更新2026-03-21 收录
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X-Ray structure of Human Deoxycytidine Kinase in complex with an inhibitor Descriptor: 4-(1-benzothiophen-2-yl)-6-[4-(2-oxo-2-pyrrolidin-1-ylethyl)piperazin-1-yl]pyrimidine, D-MALATE, Deoxycytidine kinase Authors: Tari, L.W, Swanson, R.V, Hunter, M, Hoffman, I, Stouch, T.R, Carson, K.G. Deposit date: 2009-08-18 Release date: 2010-08-18 Last modified: 2023-09-06 Method: X-RAY DIFFRACTION (2.54 Å) Cite: Lead optimization and structure-based design of potent and bioavailable deoxycytidine kinase inhibitors. Bioorg.Med.Chem.Lett., 19, 2009
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2009-08-18
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