Crystal structure of human glutaminase C in complex with the inhibitor UPGL-00019
收藏Protein Data Bank Japan2023-09-27 更新2026-03-21 收录
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Crystal structure of human glutaminase C in complex with the inhibitor UPGL-00019 Descriptor: 2-phenyl-N-{5-[4-({5-[(phenylacetyl)amino]-1,3,4-thiadiazol-2-yl}oxy)piperidin-1-yl]-1,3,4-thiadiazol-2-yl}acetamide, Glutaminase kidney isoform, mitochondrial Authors: Huang, Q, Cerione, R. Deposit date: 2016-02-19 Release date: 2016-05-11 Last modified: 2023-09-27 Method: X-RAY DIFFRACTION (2.983 Å) Cite: Design and evaluation of novel glutaminase inhibitors. Bioorg.Med.Chem., 24, 2016
创建时间:
2016-02-19



