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CASPASE2 IN COMPLEX WITH CHDI LIGAND 33c

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Protein Data Bank Japan2023-12-06 更新2026-03-21 收录
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CASPASE2 IN COMPLEX WITH CHDI LIGAND 33c Descriptor: Caspase-2, Peptide inhibitor (ACE)VDV(3PX)D-CHO Authors: Abendroth, J, Lorimer, D, Stewart, L, Maillard, M, Kiselyov, A.S. Deposit date: 2011-04-15 Release date: 2011-09-21 Last modified: 2023-12-06 Method: X-RAY DIFFRACTION (2.55 Å) Cite: Exploiting differences in caspase-2 and -3 S(2) subsites for selectivity: Structure-based design, solid-phase synthesis and in vitro activity of novel substrate-based caspase-2 inhibitors. Bioorg.Med.Chem., 19, 2011
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2011-04-15
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