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Structure of ARG1 complex with pyrrolidine-based non-boronic acid inhibitor 6

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Protein Data Bank Japan2023-10-25 更新2026-04-25 收录
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Structure of ARG1 complex with pyrrolidine-based non-boronic acid inhibitor 6 Descriptor: 1-{[(3S,4S)-3-({4-[2-(4-fluorobenzene-1-sulfonyl)ethyl]piperidin-1-yl}methyl)-4-(3-fluorophenyl)pyrrolidin-1-yl]methyl}cyclopentane-1-carboxylic acid, Arginase-1, MANGANESE (II) ION Authors: Palte, R.L, Gathiaka, S. Deposit date: 2022-08-22 Release date: 2023-03-08 Last modified: 2023-10-25 Method: X-RAY DIFFRACTION (1.84 Å) Cite: Discovery of non-boronic acid Arginase 1 inhibitors through virtual screening and biophysical methods. Bioorg.Med.Chem.Lett., 84, 2023
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2022-08-22
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