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Human neuropilin-1 in a complex with a quinoline based antagonists

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Protein Data Bank Japan2025-12-10 更新2026-04-19 收录
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Human neuropilin-1 in a complex with a quinoline based antagonists Descriptor: (2~{S})-2-[[3-[[6-[3-(aminomethyl)phenyl]quinolin-8-yl]sulfonylamino]thiophen-2-yl]carbonylamino]-5-carbamimidamido-pentanoic acid, Neuropilin-1 Authors: Djordjevic, S, Selwood, D, Hubbard, P, Leonard, P, Mota, F. Deposit date: 2024-04-30 Release date: 2025-05-14 Last modified: 2025-12-10 Method: X-RAY DIFFRACTION (1.57 Å) Cite: Quinoline-Based Neuropilin‐1 Antagonists Exhibit a Pure Antagonist Profile and Block Vascular Endothelial Growth Factor-Induced Pain. Acs Pharmacol Transl Sci, 8, 2025
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2024-04-30
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